Smartox 品牌
代理商厂商性质
北京市所在地
ω-Conotoxin-SO3 (ω-漏斗网蛛毒素SO3 )
面议ω-Conotoxin MVIIC / Omega conotoxin MVIIC (ω-漏斗网蛛毒
面议ω-Conotoxin MVIIA (ω-漏斗网蛛毒素MVIIA)
面议ω-conotoxin GVIA(ω-漏斗网蛛毒素GVIA)
面议ω-agatoxin IVA(ω-漏斗网蛛毒素 IVA)
面议Margatoxin(MgTx,玛格斑蝎毒素)
面议Kaliotoxin-1(卡利蝎毒素-1)
面议Jingzhaotoxin III(JZTx-III,敬钊缨毛蛛毒素-III)
面议Iberiotoxin 伊比(利亚)蝎毒素
面议Huwentoxin-IV(虎纹捕鸟蛛神经毒素-IV)
面议Huwentoxin-I(虎纹捕鸟蛛神经毒素-I)
面议Hainantoxin-IV(海南捕鸟蛛毒素-IV)
面议Rho-conotoxin TIA (Rho -芋螺毒素TIA )
Blocker of α1-adrenoreceptor(肾上腺素受体α1阻断剂)
Rho-conotoxin TIA has been isolated from the venom of the fish-hunting marine cone snail Conus tulipa. Rho-conotoxin TIA is a selective antagonist of α1-adrenoreceptor (α1A-, α1B- and α1D-AR). It acts non-competitively ontoα1B-adrenoreceptor but competitively on α1A-adrenoreceptor and α1D-adrenoreceptor. The most important residue for activity is Arg4. Rho-conotoxin TIA is 10-fold selective for human α1B-adrenoreceptor over
α1A-adrenoreceptor and α1D-adrenoreceptor. The IC50 values for Rho-conotoxin TIA for inhibition of 125I-BE were 18 nM for human α1A-AR, 2 nM for α1B-AR and 25 nM for α1D-AR.
Rho-conotoxin TIA 技术资料
氨基酸序列:Phe-Asn-Trp-Arg-Cys5-Cys6-Leu-Ile-Pro-Ala-Cys11-Arg-Arg-Asn-His-Lys-Lys-Phe-Cys19-NH2
二硫键: Cys5-Cys11 and Cys6-Cys19
长度 (aa):19
分子式:C105H160N36O21S4
分子量: 2390.90 Da
外观: White lyophilized solid
可溶性:aqueous buffer
CAS 号: not available
来源: Synthetic
纯度:> 97 %
产品信息
CON022-00100 | Rho-conotoxin TIA | 0.1mg |
CON022-00500 | Rho-conotoxin TIA | 0.5mg |
CON022-01000 | Rho-conotoxin TIA | 1mg |