Smartox 品牌
代理商厂商性质
北京市所在地
softwell(柔软、有弹性)细胞培养器皿
面议干细胞因子微球(StemBeads)
面议Bicolor’s Purple-Jelley Assay(透明质酸检测试剂盒)
面议Aurion 胶体金溶液(Gold Sols)
面议LudgerTag V-tag 糖肽标记和释放试剂盒
面议免疫球蛋白IgG糖基化检测/分析试剂盒——Ludger品牌
面议抗体糖基化检测/分析试剂盒——Ludger品牌
面议单克隆抗体(单抗)糖基化检测/分析试剂盒-Ludger品牌
面议弹性150mm培养皿Petrisoft-150mm dish-Non Activated-xx pK
面议弹性100mm培养皿Petrisoft-100mm dish-Non Activated-xx pK
面议弹性35mm培养皿Petrisoft-35mm dish-Non Activated-xx pKa
面议弹性150mm培养皿Petrisoft-150mm dish-Collagen I-xx pKa
面议
Tertiapin has been isolated from the venom of the Honeybee Apis mellifera. Tertiapin-Q is an oxidation-resistant mutant of the wild-type tertiapin where Methionine 13 has been replaced by a Glutamine. blocks the inwardly rectifying Kir1.1 (ROMK1) and Kir3.1/3.4 (GIRK1/GIRK4 also known as IKACh) potassium channels with Kd values of around 2 nM and 8 nM respectively. also inhibits calcium-activated large conductance BK potassium channels (KCa1.1) in a concentration and voltage-dependent manner (IC50 ~ 5 nM), in addition to inhibiting Kir3.1/3.2 (GIRK1/GIRK2) heteromultimer potassium channels with a Kd close to 270 nM. can prevent dose-dependent acetylcholine(ACh)-induced atrioventricular blocks in mammalian hearts, as KCNJ3/KCNJ5 channels (also named I(KACh)), are activated by ACh found in mammalian myocytes.
技术资料
氨基酸序列:
Ala-Leu-Cys3-Asn-Cys5-Asn-Arg-Ile-Ile-Ile-Pro-His-Gln-Cys14-Trp-Lys-Lys-Cys18-Gly-Lys-Lys-NH2
二硫键: Cys3-Cys14 and Cys5-Cys18
长度 (aa):21
分子式: C106H175N35O24S4
分子量: 2452 Da
外观:White lyophilized solid
可溶性: water and saline buffer
CAS 号: [252198-49-5]
来源: Synthetic
纯度: > 97 %
产品信息
08TER001-00100 | Tertiapin Q | 0.1mg |
08TER001-00500 | Tertiapin Q | 0.5mg |
08TER001-01000 | Tertiapin Q | 1mg |